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Search Results for " bacterial ribosome "

20

Compounds

Cat No. Product Name Synonyms Targets
T1160 Fusidic acid Fusidine Others , CAT , Antibacterial , Antibiotic
Fusidic acid (Fusidine) is an antibiotic isolated from the fermentation broth of Fusidium coccineum.
T12540 Pristinamycin IA Mikamycin IA,Mikamycin B Others , Antibiotic , P-gp
Pristinamycin IA (Mikamycin B) is a substrate for the P-glycoprotein and a cyclo-peptidic macrolactone antibiotic.
T4267 Tulathromycin A CP 472295,Draxxin,Tulathromycin Antibacterial , Antibiotic
Tulathromycin A (CP 472295) is a macrolide antibiotic.
T0788 Spectinomycin dihydrochloride Spectinomycin 2HCl,Actinospectacin ribosome , Antibacterial , Antibiotic
Spectinomycin dihydrochloride (Actinospectacin) is an antibiotic produced by Streptomyces spectabilis. It is active against gram-negative bacteria and used for the treatment of gonorrhea.
T0788L Spectinomycin dihydrochloride pentahydrate Trobicin,Spectogard,Spectinomycin hydrochloride hydrate ribosome , Antibacterial , Antibiotic
Spectinomycin dihydrochloride pentahydrate (Spectogard) is an antibiotic produced by Streptomyces spectabilis. It is active against gram-negative bacteria and used for the treatment of gonorrhea.
T1289 Fusidic acid sodium salt Sodium fusidate,Fusidate Sodium,Fucidin,SQ-16360 Others , CAT , Antibacterial , Antibiotic
Fusidic acid sodium salt (SQ-16360) is a sodium salt form of fusidic acid, a bacteriostatic antibiotic derived from the fungus Fusidium coccineum and used as a topical medication to treat skin infections.
T13767 MBX-4132 Others , Antibacterial
MBX-4132, inhibit trans translation by binding to the bacterial ribosome,is a member of a chemical class called oxadiazoles.
T6447 Clindamycin Clinimycin,Sobelin,Chlolincocin Antibacterial , Antibiotic
Clindamycin (Sobelin) dissociates peptidyl-tRNA from the bacterial ribosome, thereby disrupting bacterial protein synthesis. Clindamycin is a semisynthetic broad-spectrum antibiotic produced by chemical modification of t...
T3265 Azathramycin Desmethyl Azithromycin,6-Demethylazithromycin,Azaerythromycin A,Azaerythromycin Antibacterial , Antibiotic
Azathramycin (Desmethyl Azithromycin) is an antibiotic derived from erythromycin, binding to the 50S subunit of the bacterial ribosome, and thus inhibits translation of mRNA.
T1747 Tedizolid TR 700,DA-7157,Torezolid MAO , Antibacterial , Antibiotic
Tedizolid (DA-7157)is a novel oxazolidinone-class antibiotic that inhibits bacterial protein synthesis by binding to the 23S ribosomal RNA of the 50S subunit of the ribosome.
T5189 Omadacycline PTK 0796,Amadacycline ribosome , Antibacterial , Antibiotic
Omadacycline (Amadacycline), a new tetracycline antibiotic, can inhibit the 30s subunit of bacterial ribosome.
T11836 Lefamulin acetate BC-3781 acetate ribosome , Antibacterial , Antibiotic
Lefamulin acetate (BC-3781 acetate) (formally BC-3781 acetate) is a novel pleuromutilin antibiotic and is the first to be used for the systemic treatment of bacterial infections in humans. Lefamulin acetate (BC-3781 acet...
T0912 Tetracycline hydrochloride NCI-c55561,Tetracycline HCl ribosome , Antibacterial , Antibiotic
Tetracycline hydrochloride (NCI-c55561) is the hydrochloride salt of the tetracycline, a broad-spectrum naphthacene antibiotic produced semisynthetically from chlortetracycline, an antibiotic isolated from the bacterium ...
T71810 Thiamphenicol palmitate
Thiamphenicol palmitate is a Prodrug of Thiamphenicol, inhibiting the 50S subunit of the bacterial ribosome and protein translation.
T11842 Levomecol Others
Levomecol, a broad-spectrum antibiotic derived from Streptomyces venezuelae, comprises Chloramphenicol and Methyluracil. It exerts its bacteriostatic effect by binding to the bacterial ribosome, inhibiting protein synthe...
T70076 NOSO-95C
NOSO-95C is an antibacterial compound that bind to the bacterial ribosome and kill bacteria through inhibition of the translation. NOSO-95C showed promising in vitro and in vivo efficacy against Enterobacteriaceae.
T70250 Demeclocycline calcium
Demeclocycline calcium is a semisynthetic tetracycline antibiotic which was derived from a strain of Streptomyces aureofaciens. Demeclocycline binds to bacterial 30S ribosomal subunit and prevents binding of aminoacyl-tR...
T60300 BPH-1086
BPH-1086 (compound 10) is an inhibitor of IspH. IspH domain fused with ribosomal protein S1 (RPS1) can bind to mRNA or form part of the bacterial ribosome [1] [2].
T79015 SEQ-9
SEQ-9 is an orally active inhibitor targeting the Mycobacterium tuberculosis (Mtb) 23S bacterial ribosome, demonstrating an inhibitory concentration (IC50) around 170 nM against unmethylated Mtb ribosomes and showing pot...
T75318 Spectinomycin
Spectinomycin, a broad-spectrum antibiotic, targets and inhibits the growth of various gram-positive and gram-negative organisms by selectively binding to the bacterial ribosome, disrupting protein synthesis. Additionall...

Compounds

Fusidic acid
T1160
Synonym: Fusidine
Target: Others, CAT, Antibacterial, Antibiotic
Pristinamycin IA
T12540
Synonym: Mikamycin IA,Mikamycin B
Target: Others, Antibiotic, P-gp
Tulathromycin A
T4267
Synonym: CP 472295,Draxxin,Tulathromycin
Target: Antibacterial, Antibiotic
Spectinomycin dihydrochloride
T0788
Synonym: Spectinomycin 2HCl,Actinospectacin
Target: ribosome, Antibacterial, Antibiotic
Spectinomycin dihydrochloride pentahydrate
T0788L
Synonym: Trobicin,Spectogard,Spectinomycin hydrochloride hydrate
Target: ribosome, Antibacterial, Antibiotic
Fusidic acid sodium salt
T1289
Synonym: Sodium fusidate,Fusidate Sodium,Fucidin,SQ-16360
Target: Others, CAT, Antibacterial, Antibiotic
MBX-4132
T13767
Synonym:
Target: Others, Antibacterial
Clindamycin
T6447
Synonym: Clinimycin,Sobelin,Chlolincocin
Target: Antibacterial, Antibiotic
Azathramycin
T3265
Synonym: Desmethyl Azithromycin,6-Demethylazithromycin,Azaerythromycin A,Azaerythromycin
Target: Antibacterial, Antibiotic
Tedizolid
T1747
Synonym: TR 700,DA-7157,Torezolid
Target: MAO, Antibacterial, Antibiotic
Omadacycline
T5189
Synonym: PTK 0796,Amadacycline
Target: ribosome, Antibacterial, Antibiotic
Lefamulin acetate
T11836
Synonym: BC-3781 acetate
Target: ribosome, Antibacterial, Antibiotic
Tetracycline hydrochloride
T0912
Synonym: NCI-c55561,Tetracycline HCl
Target: ribosome, Antibacterial, Antibiotic
Thiamphenicol palmitate
T71810
Synonym:
Target:
Levomecol
T11842
Synonym:
Target: Others
NOSO-95C
T70076
Synonym:
Target:
Demeclocycline calcium
T70250
Synonym:
Target:
BPH-1086
T60300
Synonym:
Target:
SEQ-9
T79015
Synonym:
Target:
Spectinomycin
T75318
Synonym:
Target:
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TargetMol